SCHEMBL20049293

SCHEMBL20049293

CCc1cc(F)c2nc(C)cnc2c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.33
HRH4 Q9H3N8 2/20 0.33
HRH3 Q9Y5N1 2/20 0.33
HRH2 P25021 1/20 0.31
HRH1 P35367 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20049119 0.83 KCNH2 (0.34) KCNH2HRH4HRH3HRH2HRH1
SCHEMBL20048949 0.73 KCNH2 (0.31) KCNH2HRH4HRH3
SCHEMBL20675598 0.71 CCR1 (0.46) KCNH2
Ethoxycarbonyl Group SCHEMBL28040584 0.71
SCHEMBL20049379 0.71
SCHEMBL30900020 0.70 NPC1 (0.41) HRH4
SCHEMBL20049186 0.70 NPC1 (0.41) HRH4
SCHEMBL103875 0.66 ALDH1A1 (0.42) CYP11B1CYP11B2
SCHEMBL24019244 0.66 HSD17B10 (0.34)
SCHEMBL18876144 0.66 MEN1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067704-A1 ISOXAZOLE ANALOGS AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2018-04-12 WO disclosed