SCHEMBL20049296

SCHEMBL20049296

Cc1cnc2cc(C(C)C)cc(Cl)c2n1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
NR4A2 P43354 2/20 0.31
KCNH2 Q12809 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20048949 0.80 KCNH2 (0.31) KCNH2HRH4HRH3
SCHEMBL20675596 0.72 CCR1 (0.43) MAPTRAB9APDE2APDE10ANR4A2
SCHEMBL20666234 0.71 NR4A2 (0.41) ALDH1A1LMNAMAPTSMN1; SMN2NR4A2
SCHEMBL20675602 0.71 CCR1 (0.46)
SCHEMBL20049295 0.70 NPC1 (0.41) ALDH1A1NPC1LMNAMAPTRAB9A
SCHEMBL14652456 0.70 NPC1 (0.41) ALDH1A1NPC1LMNAMAPTRAB9A
SCHEMBL24009618 0.68 ALDH1A1 (0.41) ALDH1A1LMNASMN1; SMN2
SCHEMBL7451226 0.68 NR4A2 (0.46) ALDH1A1NR4A2
SCHEMBL20666241 0.68 EGFR (0.30)
SCHEMBL24019234 0.68 OGA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018067704-A1 ISOXAZOLE ANALOGS AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2018-04-12 WO disclosed