SCHEMBL20051525

SCHEMBL20051525

N#CN1CCCC(C(=O)Nc2ncc(-c3ccccc3)s2)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 16/20 1.00
UCHL1 P09936 2/20 0.88
MKNK1 Q9BUB5 1/20 0.62
OTUD7B Q6GQQ9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23198226 1.00 USP30 (1.00) USP30UCHL1MKNK1OTUD7B
SCHEMBL23198203 1.00 USP30 (1.00) USP30UCHL1MKNK1OTUD7B
SCHEMBL17632033 0.94 UCHL1 (1.00) USP30UCHL1MKNK1OTUD7B
SCHEMBL17632038 0.94 UCHL1 (1.00) USP30UCHL1MKNK1OTUD7B
SCHEMBL23403455 0.87 UCHL1 (0.87) USP30UCHL1MKNK1OTUD7B
SCHEMBL17632208 0.87 UCHL1 (0.87) USP30UCHL1MKNK1OTUD7B
SCHEMBL17632501 0.85 UCHL1 (0.83) USP30UCHL1MKNK1OTUD7B
SCHEMBL29992744 0.85 UCHL1 (0.83) USP30UCHL1MKNK1OTUD7B
SCHEMBL17631603 0.84 UCHL1 (0.83) USP30UCHL1MKNK1OTUD7B
SCHEMBL17631683 0.84 UCHL1 (0.83) USP30UCHL1MKNK1OTUD7B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109803963-B Cyano-substituted heterocycles having USP30 inhibitor activity 特殊治疗有限公司 2022-04-26 CN claimed
CN-109803963-B Cyano-substituted heterocycles having USP30 inhibitor activity 特殊治疗有限公司 2022-04-26 CN disclosed
EP-3523291-B1 CYANO-SUBSTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LTD (GB) 2021-04-14 EP disclosed
WO-2018065768-A1 CYANO-SUBSTITUTED HETEROCYCLES WITH ACTIVITY AS INHIBITORS OF USP30 MISSION THERAPEUTICS LIMITED (GB) 2018-04-12 WO disclosed