SCHEMBL20052428

SCHEMBL20052428

Cn1cc(C[C@H](NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)OCc2ccccc2)C(=O)NCC(=O)N[C@H](/C=C/S(C)(=O)=O)CC(=O)OC(C)(C)C)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 15/20 0.51
CASP7 P55210 10/20 0.49
CASP1 P29466 7/20 0.49
PSMB5 P28074 3/20 0.48
CASP9 P55211 4/20 0.45
CASP4 P49662 3/20 0.44
CASP5 P51878 2/20 0.44
CASP8 Q14790 2/20 0.44
CASP10 Q92851 2/20 0.44
CASP2 P42575 1/20 0.44
CASP6 P55212 1/20 0.43
CCKAR P32238 2/20 0.43
CCKBR P32239 2/20 0.43
OPRD1 P41143 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19944808 0.91 PSMB5 (0.49) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL20052456 0.91 CASP3 (0.62) CASP3CASP7CASP1CASP9CASP4
SCHEMBL15462695 0.90 CASP3 (0.65) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL20355913 0.90 CASP3 (0.65) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL20355912 0.90 CASP3 (0.65) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL20052371 0.90 CASP3 (0.65) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL19015746 0.84 CASP3 (0.59) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL20052427 0.84 CASP3 (0.61) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL19015922 0.82 CASP3 (0.61) CASP3CASP7CASP1PSMB5CASP9
SCHEMBL18782201 0.82 CASP3 (0.61) CASP3CASP7CASP1PSMB5CASP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9944674-B2 Selective cysteine protease inhibitors and uses thereof GENESIS TECHNOLOGIES LIMITED (BB) 2018-04-17 US disclosed