SCHEMBL20054426

SCHEMBL20054426

O=C(NCc1nc2c([nH]1)-c1ccc(-c3ccc4c(ccc5nc(CNC(=O)C6CCC(F)(F)CC6)[nH]c54)c3)cc1CC2)C1CCC(F)(F)CC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 12/20 0.37
DYRK1A Q13627 10/20 0.37
WNT1 P04628 8/20 0.35
PDPK1 O15530 2/20 0.32
JAK1 P23458 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
KCNH2 Q12809 1/20 0.31
MAP4K1 Q92918 1/20 0.31
PARP1 P09874 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20054516 0.89 GSK3B (0.40) GSK3BDYRK1AWNT1PDPK1JAK1
SCHEMBL20054506 0.88 GSK3B (0.45) GSK3BDYRK1AWNT1PDPK1JAK1
SCHEMBL20054378 0.83 GSK3B (0.37) GSK3BDYRK1AWNT1JAK1HTR1A
SCHEMBL20054417 0.80 GSK3B (0.49) GSK3BDYRK1AWNT1PDPK1
SCHEMBL15116591 0.79 GSK3B (0.36) GSK3BDYRK1AWNT1PDPK1MAP4K1
SCHEMBL19388329 0.79 GSK3B (0.36) GSK3BDYRK1AWNT1PDPK1MAP4K1
SCHEMBL20054459 0.76
SCHEMBL20221280 0.75 GSK3B (0.37) GSK3BDYRK1AWNT1PDPK1JAK1
SCHEMBL20054351 0.73 GSK3B (0.43) GSK3BDYRK1AWNT1PDPK1HTR1A
SCHEMBL19883180 0.70 MPL (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed