SCHEMBL20054516

SCHEMBL20054516

O=C(NCc1nc2c([nH]1)-c1ccc(-c3ccc4c(c3)CCc3nc(CNC(=O)C5CCC(F)(F)CC5)[nH]c3-4)cc1CC2)C1CCC(F)(F)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.40
DYRK1A Q13627 10/20 0.40
WNT1 P04628 8/20 0.38
HTR1A P08908 2/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
KCNH2 Q12809 2/20 0.36
JAK1 P23458 1/20 0.35
MAPK14 Q16539 2/20 0.34
GSK3A P49840 1/20 0.34
PDPK1 O15530 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20054378 0.92 GSK3B (0.37) GSK3BDYRK1AWNT1HTR1ADRD2
SCHEMBL20054426 0.89 GSK3B (0.37) GSK3BDYRK1AWNT1HTR1ADRD2
SCHEMBL19388305 0.77 GSK3B (0.39) GSK3BDYRK1AWNT1KCNH2PDPK1
SCHEMBL15116588 0.77 GSK3B (0.39) GSK3BDYRK1AWNT1KCNH2PDPK1
SCHEMBL20054505 0.76
SCHEMBL20054351 0.76 GSK3B (0.43) GSK3BDYRK1AWNT1HTR1ADRD2
SCHEMBL20054506 0.73 GSK3B (0.45) GSK3BDYRK1AWNT1HTR1ADRD2
SCHEMBL20054480 0.72 GSK3B (0.61) GSK3BDYRK1AWNT1
SCHEMBL15116781 0.71 GSK3B (0.36) GSK3BDYRK1AWNT1KCNH2
SCHEMBL19388310 0.71 GSK3B (0.36) GSK3BDYRK1AWNT1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed