SCHEMBL20054467

SCHEMBL20054467

NCc1ncc(-c2ccc(-c3ccc(-c4cnc(CN)[nH]4)s3)cc2)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.40
SCN10A Q9Y5Y9 8/20 0.39
SCN5A Q14524 2/20 0.39
APP P05067 1/20 0.36
KLK1 P06870 1/20 0.36
KLK5 Q9Y337 1/20 0.36
ASIC3 Q9UHC3 1/20 0.35
CYP2E1 P05181 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
MASP2 O00187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20055405 0.77 TRPV1 (0.46) PDE10ASCN10ASCN5AMASP2
SCHEMBL2562957 0.76 PDE10A (0.64) PDE10AKLK1KLK5MASP2
SCHEMBL25303515 0.73 SCN2A (0.55) PDE10ASCN10ASCN5A
SCHEMBL12648128 0.73 NLN (0.41) PDE10ASCN10ASCN5A
SCHEMBL19388645 0.73 SCN10A (0.40) SCN10ASCN5A
SCHEMBL15114359 0.73 SCN10A (0.40) SCN10ASCN5A
SCHEMBL20054552 0.72 NLN (0.43) PDE10ASCN10ASCN5A
Bromide SCHEMBL16210189 0.72 SCN2A (0.54) PDE10ASCN10ASCN5A
Bromide SCHEMBL25307759 0.72 SCN10A (0.56) SCN10ASCN5A
SCHEMBL20054471 0.71 NLN (0.42) PDE10ASCN10ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019196-B1 COMBINATIONS OF HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-06-06 EP disclosed
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed