SCHEMBL20054545

SCHEMBL20054545

CC(C)(C)OC(=O)NC(c1nc2ccc(-c3ccc(-c4ccc5nc(C(NC(=O)OC(C)(C)C)C(C)(C)C)[nH]c5c4)cc3)cc2[nH]1)C(C)(C)C

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 10/20 0.64
SCN10A Q9Y5Y9 3/20 0.42
MLKL Q8NB16 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
LCK P06239 1/20 0.40
MAP4K4 O95819 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15116826 1.00 AAK1 (0.64) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL15116825 0.93 AAK1 (0.57) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL20054463 0.93 AAK1 (0.57) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL15116865 0.91 AAK1 (0.55) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL15116803 0.91 AAK1 (0.55) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL20054558 0.91 AAK1 (0.55) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL20054464 0.88 AAK1 (0.52) AAK1SCN10AMLKLTRPV1
SCHEMBL15116827 0.88 AAK1 (0.52) AAK1SCN10AMLKLTRPV1
SCHEMBL15116772 0.87 AAK1 (0.66) AAK1SCN10AMLKLTRPV1LCK
SCHEMBL15116746 0.87 AAK1 (0.50) AAK1SCN10ALCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2802326-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-04-18 EP disclosed