SCHEMBL20056946

SCHEMBL20056946

Cc1cnn(Cc2ccc(CN=O)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 17/20 0.49
KLK1 P06870 1/20 0.43
HSD17B10 Q99714 1/20 0.42
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15759268 0.84 KLKB1 (0.51) KLKB1KLK1HSD17B10ALDH1A1
SCHEMBL16246747 0.81 KLKB1 (0.49) KLKB1KLK1HSD17B10
SCHEMBL13813853 0.81 KCNH2 (0.53) KLKB1HSD17B10ALDH1A1
SCHEMBL17232474 0.81 KLKB1 (0.49) KLKB1KLK1HSD17B10
SCHEMBL15033959 0.79 KLKB1 (0.51) KLKB1KLK1HSD17B10
SCHEMBL13102481 0.79 KLKB1 (0.54) KLKB1KLK1
SCHEMBL16246702 0.79 KLKB1 (0.48) KLKB1KLK1HSD17B10ALDH1A1
SCHEMBL27239076 0.79 KLKB1 (0.65) KLKB1KLK1
SCHEMBL130830 0.79 L3MBTL1 (0.62) KLKB1ALDH1A1POLB
SCHEMBL16486803 0.79 KLKB1 (0.48) KLKB1KLK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309152-A1 ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE Vertex Pharmaceuticals Incorporated (US) 2018-04-18 EP disclosed