SCHEMBL20060246

SCHEMBL20060246

COc1cc(OCCN2CCCC2)ccc1C

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.60
TDP1 Q9NUW8 1/20 0.57
LTA4H P09960 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
HTT P42858 2/20 0.57
POLB P06746 1/20 0.56
ALDH1A1 P00352 1/20 0.52
MAOB P27338 1/20 0.52
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
PSMB1 P20618 1/20 0.51
PSMB5 P28074 1/20 0.51
PSMB2 P49721 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13849416 0.99 KDM4E (0.59) KDM4ETDP1LTA4HSMN1; SMN2HTT
SCHEMBL1911862 0.90 MEN1 (0.53) KDM4ELTA4HSMN1; SMN2ALDH1A1
SCHEMBL1911850 0.87 NPC1 (0.66) KDM4ESMN1; SMN2POLBALDH1A1
SCHEMBL13849370 0.87 SMN1; SMN2 (0.63) KDM4ELTA4HSMN1; SMN2HTTPOLB
SCHEMBL12961350 0.86 DRD3 (0.47) KDM4ETDP1LTA4HSMN1; SMN2HTT
SCHEMBL13849419 0.85 KDM4E (0.51) KDM4ESMN1; SMN2HTTMAOB
SCHEMBL13849420 0.85 MAOB (0.50) KDM4ELTA4HALDH1A1MAOBESR1
SCHEMBL13091445 0.84 KDM4E (0.71) KDM4ELTA4HSMN1; SMN2HTTALDH1A1
SCHEMBL1964263 0.84 LTA4H (0.59) KDM4ELTA4HSMN1; SMN2POLBALDH1A1
SCHEMBL1962645 0.83 LTA4H (0.58) KDM4ELTA4HPOLBPSMB1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595987-B1 NEW AMINOPYRAZOLOQUINAZOLINES BOEHRINGER INGELHEIM INT (DE) 2018-04-18 EP disclosed