SCHEMBL20064607

SCHEMBL20064607

C=CCc1ccc(OC(F)F)c(O[C@H]2C[C@H](C(=O)N[C@H]3CC[C@H](C(C)(O)C(F)(F)F)CC3)C2)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
PDE4D Q08499 8/20 0.35
PDE4A P27815 6/20 0.35
PDE4B Q07343 5/20 0.35
PDE4C Q08493 5/20 0.35
PPARA Q07869 1/20 0.34
HPGDS O60760 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PTGS1 P23219 1/20 0.32
KCNH2 Q12809 1/20 0.32
PTGES O14684 1/20 0.32
CTSD P07339 1/20 0.32
ENPP2 Q13822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21222484 0.85 PDE4D (0.38) MEN1KMT2APDE4DPDE4APDE4B
SCHEMBL21222480 0.85 PDE4D (0.38) MEN1KMT2APDE4DPDE4APDE4B
SCHEMBL21227930 0.85 PDE4D (0.38) MEN1KMT2APDE4DPDE4APDE4B
SCHEMBL20064509 0.83 NPC1 (0.50) MEN1NPC1RAB9AKMT2APPARA
SCHEMBL20065559 0.79 NPC1 (0.41) MEN1NPC1RAB9AKMT2APPARA
SCHEMBL21222653 0.77 HPGDS (0.44) MEN1KMT2APDE4DPDE4APDE4B
SCHEMBL21222656 0.77 HPGDS (0.44) MEN1KMT2APDE4DPDE4APDE4B
SCHEMBL21221974 0.76 HPGDS (0.44) KMT2APDE4DPDE4APDE4BPDE4C
SCHEMBL20065702 0.76 HPGDS (0.44) KMT2APDE4DPDE4APDE4BPDE4C
SCHEMBL21221977 0.75 HPGDS (0.45) MEN1KMT2APDE4DPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018069863-A1 1,3 DI-SUBSTITUTED CYCLOBUTANE OR AZETIDINE DERIVATIVES AS HEMATOPOIETIC PROSTAGLANDIN D SYNTHASE INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-04-19 WO disclosed