SCHEMBL20071863

SCHEMBL20071863

CN(C)C(=O)c1ccc(N2CCC(C)(C)CC2)nc1Cl

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 2/20 0.39
CNR2 P34972 1/20 0.35
CNR1 P21554 1/20 0.34
HSD11B1 P28845 1/20 0.34
DGAT1 O75907 1/20 0.34
KCNH2 Q12809 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KIF18A Q8NI77 2/20 0.32
PARP1 P09874 1/20 0.32
TPH1 P17752 1/20 0.32
SMO Q99835 1/20 0.32
CHRM4 P08173 1/20 0.32
ADRB2 P07550 1/20 0.32
MAPK1 P28482 1/20 0.31
OGA O60502 1/20 0.31
PTPN11 Q06124 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20071864 0.88 PTPN11 (0.41) PTGER4CNR2CNR1HSD11B1PIK3C3
SCHEMBL20071865 0.84 PTGER4 (0.32) PTGER4CNR1HSD11B1TPH1SMO
SCHEMBL21644403 0.83 PTGER4 (0.32) PTGER4HSD11B1TPH1MAPK1PTPN11
SCHEMBL20072210 0.82 ALDH1A1 (0.39) HSD11B1ALDH1A1SMONR1H2NR1H3
SCHEMBL20072195 0.82 PTGER4 (0.44) PTGER4CNR1HSD11B1SMOPTPN11
SCHEMBL23838140 0.82 NR1H2 (0.42) PTGER4CNR1PARP1SMONR1H2
SCHEMBL21644381 0.81 PTGER4 (0.33) PTGER4PTPN11
SCHEMBL23838054 0.81 DYRK1A (0.33) PTGER4KIF18APARP1TPH1SMO
SCHEMBL23838145 0.80 NR1H2 (0.41) PTGER4CNR2CNR1HSD11B1ALDH1A1
SCHEMBL23838112 0.80 PTGER4 (0.30) PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018068297-A1 N-ARYL AND N-HETEROARYL PIPERIDINE DERIVATIVES AS LIVER X RECEPTOR β AGONISTS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2018-04-19 WO disclosed