SCHEMBL2007198

SCHEMBL2007198

Cc1c(CC(=O)O)c2cc(O)c(F)cc2n1C(=O)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
NFKB1 P19838 1/20 0.45
HIF1A Q16665 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
AKR1C3 P42330 4/20 0.44
AKR1C2 P52895 4/20 0.44
PTGDR2 Q9Y5Y4 8/20 0.43
CCKAR P32238 1/20 0.43
PTGS1 P23219 3/20 0.43
PTGS2 P35354 3/20 0.43
ABCB1 P08183 1/20 0.43
PTGDR Q13258 1/20 0.41
HSD17B14 Q9BPX1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006767 0.88 PTGS1 (0.49) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL2004590 0.87 PTGS1 (0.52) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3001769 0.85 LMNA (0.61) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL2008114 0.84 PTGS1 (0.61) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL2001676 0.82 LMNA (0.39) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL2009264 0.82 AKR1C3 (0.54) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL2002636 0.80 AKR1C3 (0.49) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL5439139 0.79 AKR1C3 (0.62) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL5443931 0.79 PTGS1 (0.64) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL5447453 0.79 AKR1C3 (0.66) LMNACYP1A2CYP2D6CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed