SCHEMBL20073552

SCHEMBL20073552

CCc1ccc(N)c(N(C)S(C)(=O)=O)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 14/20 0.42
CA2 P00918 1/20 0.38
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.36
PARP1 P09874 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29739879 1.00 CYP19A1 (0.42) CYP19A1CA2HPGDKMT2APARP1
SCHEMBL20155989 0.83 CYP19A1 (0.39) CYP19A1CA2HPGDKMT2APARP1
SCHEMBL20073408 0.83 CYP19A1 (0.45) CYP19A1CA2KMT2A
SCHEMBL24498144 0.81 PARP1 (0.39) CYP19A1HPGDKMT2APARP1ALDH1A1
SCHEMBL26544480 0.80 CYP19A1 (0.37) CYP19A1CA2HPGDKMT2APARP1
SCHEMBL26514276 0.80 CYP19A1 (0.37) CYP19A1CA2HPGDKMT2APARP1
SCHEMBL25213378 0.79 CA1 (0.44) CYP19A1CA2ALDH1A1
SCHEMBL13580500 0.78 SLC6A2 (0.40) HPGDKMT2AALDH1A1
SCHEMBL20150117 0.78 ALDH1A1 (0.37) CYP19A1HPGDKMT2APARP1ALDH1A1
SCHEMBL26512401 0.78 SLC6A2 (0.43) CYP19A1HPGDKMT2APARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240101548-A1 HYDROXAMATE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF SHENZHEN CHIPSCREEN BIOSCIENCES CO., LTD (CN) 2024-03-28 US disclosed
EP-4257587-A1 HYDROXAMATE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shenzhen Chipscreen Biosciences Co., Ltd. (CN) 2023-10-11 EP disclosed
CN-116283954-A Hydroxamate compound, preparation method and application thereof 深圳微芯生物科技股份有限公司 2023-06-23 CN disclosed
CN-114901656-B Hydroximic acid ester compound, preparation method and application thereof 深圳微芯生物科技股份有限公司 2023-04-07 CN disclosed
CN-114901656-A Hydroximic acid ester compound, preparation method and application thereof 深圳微芯生物科技股份有限公司 2022-08-12 CN disclosed
WO-2022117016-A1 HYDROXAMATE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 深圳微芯生物科技股份有限公司 2022-06-09 WO disclosed
WO-2022117016-A1 HYDROXAMATE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 深圳微芯生物科技股份有限公司 2022-06-09 WO disclosed
US-11220508-B2 TYK2 inhibitors and uses thereof NIMBUS LAKSHMI, INC. (US) 2022-01-11 US disclosed
US-11174265-B2 2021-11-16 US disclosed
EP-3848370-A2 TYK2 INHIBITORS AND USES THEREOF Nimbus Lakshmi, Inc. (US) 2021-07-14 EP disclosed
US-10323036-B2 TYK2 inhibitors and uses thereof NIMBUS LAKSHMI, INC. (US) 2019-06-18 US disclosed
US-20180155349-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-06-07 US disclosed
US-20180155349-A1 TYK2 INHIBITORS AND USES THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-06-07 US disclosed
WO-2018071794-A1 TYK2 INHIBITORS AND USES THEREOF NIMBUS LAKSHMI, INC. (US) 2018-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11220508-B2 TYK2 inhibitors and uses thereof TYK2, JAK2, JAK1 CYP19A1 2724/4885CA2 4600/4885HPGD 4476/4885
US-20240101548-A1 HYDROXAMATE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF TYK2, WEE2, WEE1 CYP19A1 1198/4885CA2 1381/4885HPGD 683/4885
US-10323036-B2 TYK2 inhibitors and uses thereof TYK2, JAK2, JAK1 CYP19A1 2724/4885CA2 4600/4885HPGD 4476/4885
US-11174265-B2 TYK2, JAK2, JAK1 CYP19A1 2529/4885CA2 4506/4885HPGD 4569/4885
US-20180155349-A1 TYK2 INHIBITORS AND USES THEREOF TYK2, JAK2, JAK1 CYP19A1 2724/4885CA2 4600/4885HPGD 4476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.