SCHEMBL20074474

SCHEMBL20074474

Cc1cccc(-c2nc3n(c2-c2ccnc(-c4ccc(C(=O)NC5CCOCC5)cc4)c2)[C@@H]2CCC3C2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 20/20 1.00
KDR P35968 10/20 1.00
MAPK14 Q16539 4/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20074390 1.00 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074404 1.00 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074398 1.00 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074414 0.86 TGFBR1 (0.85) TGFBR1KDRMAPK14
SCHEMBL20074410 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074560 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074555 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074463 0.85 TGFBR1 (1.00) TGFBR1KDRMAPK14
SCHEMBL20074460 0.82 TGFBR1 (0.80) TGFBR1KDRMAPK14
SCHEMBL5787523 0.82 TGFBR1 (0.69) TGFBR1KDRMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018068759-A1 FIVE-MEMBERED HETEROARYL RING BRIDGED RING DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 江苏恒瑞医药股份有限公司 2018-04-19 WO disclosed