SCHEMBL20074780

SCHEMBL20074780

Cn1nc(-c2ccc(C#N)cc2)c(O)c1N

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.42
MMP3 P08254 1/20 0.42
NSD2 O96028 1/20 0.41
EGLN2 Q96KS0 3/20 0.40
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
KDM4C Q9H3R0 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MAPK14 Q16539 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
HRH4 Q9H3N8 2/20 0.37
SLC34A1 Q06495 1/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20074694 0.83 CYP11B2 (0.46) CYP11B2NSD2BRAFKDRKDM4C
SCHEMBL20075467 0.79 NSD2 (0.45) CYP11B2MMP3NSD2EGLN2KDM4C
SCHEMBL20075173 0.79 SLC34A1 (0.47) CYP11B2NSD2EGLN2BRAFKDR
SCHEMBL20074777 0.79 SLC34A1 (0.47) CYP11B2NSD2BRAFKDRSLC34A1
SCHEMBL20075477 0.79 MAPK14 (0.59) BRAFKDRKDM4CMAPK14
SCHEMBL4048227 0.71 TLR7 (0.50) CYP11B2NSD2HRH3
SCHEMBL20074806 0.70 CYP11B2 (0.46) CYP11B2NSD2EGLN2KDM4CHRH3
SCHEMBL15727494 0.69 HRH4 (0.48) CYP11B2EGLN2HRH3HRH4
SCHEMBL20074788 0.69 MAPK14 (0.55) BRAFKDRMAPK14SLC34A1CA12
SCHEMBL18988210 0.69 ADORA1 (0.50) MAPK14CA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3526212-B1 SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF BAYER AG (DE) 2021-12-22 EP disclosed
WO-2018069222-A1 SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF BAYER AKTIENGESELLSCHAFT (DE) 2018-04-19 WO disclosed