SCHEMBL20078232

SCHEMBL20078232

CC(C)c1cnn(-c2cc(C(C)(C)c3cnn(-c4cccc(F)c4)c3)ccc2F)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
GRM4 Q14833 1/20 0.34
RXRA P19793 11/20 0.34
GRIN1 Q05586 11/20 0.34
GRIN2B Q13224 11/20 0.34
EPHX2 P34913 1/20 0.33
KCNT1 Q5JUK3 1/20 0.32
MTOR P42345 1/20 0.32
KAT6A Q92794 1/20 0.31
KEAP1 Q14145 1/20 0.31
NOTUM Q6P988 1/20 0.31
CASR P41180 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18878403 0.81 NPC1 (0.47) NPC1GRM4RXRAGRIN1GRIN2B
SCHEMBL21064022 0.78 RXRA (0.36) NPC1GRM4RXRAGRIN1GRIN2B
SCHEMBL26054257 0.73 NPC1 (0.47) NPC1GRM4RXRAGRIN1GRIN2B
SCHEMBL27498530 0.70 EPHX2 (0.63) NPC1RXRAGRIN1GRIN2BEPHX2
SCHEMBL2609429 0.69 RXRA (0.41) RXRAGRIN1GRIN2BMTORKAT6A
SCHEMBL25015837 0.69 EPHX2 (0.54) NPC1RXRAGRIN1GRIN2BEPHX2
SCHEMBL2609427 0.68 KDM5B (0.48) RXRAGRIN1GRIN2BKCNT1NOTUM
SCHEMBL21478371 0.68 RXRA (0.44) RXRAGRIN1GRIN2B
SCHEMBL2609426 0.68 CFTR (0.43) NPC1
SCHEMBL21146830 0.68 GCGR (0.34) RXRAGRIN1GRIN2BMTORNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9951074-B2 Dihydropteridinone derivatives and uses thereof DANA-FARBER CANCER INSTITUTE, INC. (US) 2018-04-24 US disclosed