SCHEMBL20080348

SCHEMBL20080348

CCC(=O)c1cn(-c2ccccn2)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.52
HTR3A P46098 4/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
TSHR P16473 1/20 0.47
MEN1 O00255 5/20 0.46
HTR7 P34969 2/20 0.44
POLB P06746 1/20 0.43
MITF O75030 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20080410 0.91 HTR3A (0.51) KMT2AHTR3AL3MBTL1TSHRHTR7
SCHEMBL15444633 0.86 HTR3A (0.56) KMT2AHTR3AHTR7POLBALDH1A1
SCHEMBL19969879 0.86 HTR3A (0.54) KMT2AHTR3AL3MBTL1TSHRMEN1
SCHEMBL6044056 0.83 HTR3A (0.53) HTR3AL3MBTL1TSHRHTR7POLB
SCHEMBL15440779 0.81 HTR3A (0.54) HTR3ATSHRHTR7POLBALDH1A1
SCHEMBL15420930 0.81 NR4A2 (0.64) KMT2AHTR3AL3MBTL1TSHRMEN1
SCHEMBL20080370 0.81 HTR3A (0.54) KMT2AHTR3AL3MBTL1TSHRMEN1
SCHEMBL18539469 0.80 HTR3A (0.46) KMT2AHTR3ATSHRMEN1HTR7
SCHEMBL23812575 0.80 KMT2A (0.53) KMT2AHTR3AL3MBTL1TSHRMEN1
SCHEMBL19068175 0.79 HTR3A (0.53) KMT2AHTR3AL3MBTL1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312169-B1 5-HT3 RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICALS CO (JP) 2021-09-15 EP disclosed
EP-3312169-A1 5-HT3 RECEPTOR ANTAGONISTS Takeda Pharmaceutical Company Limited (JP) 2018-04-25 EP disclosed