SCHEMBL20080419

SCHEMBL20080419

CCC(=O)c1cn(-c2cnn(C)c2)c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 12/20 0.55
KMT2A Q03164 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
TSHR P16473 1/20 0.46
NR4A2 P43354 1/20 0.45
MEN1 O00255 1/20 0.45
ENPP2 Q13822 1/20 0.44
MITF O75030 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17652247 0.87 HTR3A (0.59) HTR3ANR4A2ENPP2
SCHEMBL18922760 0.85 HTR3A (0.58) HTR3AKMT2AL3MBTL1TSHRNR4A2
SCHEMBL15444637 0.85 HTR3A (0.58) HTR3AL3MBTL1NR4A2ENPP2ALDH1A1
Hydrochloric Acid SCHEMBL15421042 0.85 HTR3A (0.58) HTR3ANR4A2ENPP2
SCHEMBL15440798 0.82 HTR3A (0.58) HTR3ATSHRNR4A2ALDH1A1
SCHEMBL15420954 0.82 NR4A2 (0.69) HTR3AKMT2AL3MBTL1TSHRNR4A2
SCHEMBL23812548 0.81 HTR3A (0.53) HTR3AKMT2AL3MBTL1TSHRNR4A2
SCHEMBL23812575 0.80 KMT2A (0.53) HTR3AKMT2AL3MBTL1TSHRNR4A2
SCHEMBL19068198 0.80 HTR3A (0.53) HTR3AKMT2AL3MBTL1TSHRNR4A2
SCHEMBL18922736 0.79 HTR3A (0.54) HTR3AKMT2AL3MBTL1TSHRNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3312169-A1 5-HT3 RECEPTOR ANTAGONISTS Takeda Pharmaceutical Company Limited (JP) 2018-04-25 EP disclosed