SCHEMBL20083706

SCHEMBL20083706

O=C(CCn1ccnc1-c1ccccc1)OCc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.67
PLAA Q9Y263 1/20 0.44
MAPK1 P28482 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALPG P10696 1/20 0.44
PDE6D O43924 2/20 0.43
LMNA P02545 1/20 0.41
BRD4 O60885 1/20 0.41
LIMK2 P53671 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
JMJD6 Q6NYC1 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4429718 0.87 ESR1 (0.70) ESR1PLAAALDH1A1CYP1A2CYP2C9
SCHEMBL5329152 0.87 ESR1 (0.55) ESR1PLAAMAPK1L3MBTL1ALDH1A1
SCHEMBL17916296 0.85 ESR1 (0.67) ESR1PLAAALDH1A1CYP2C9CYP2C19
SCHEMBL5707890 0.85 ESR1 (0.67) ESR1PLAAALDH1A1CYP2C9CYP2C19
SCHEMBL18510090 0.85 ESR1 (0.67) ESR1PLAAALDH1A1CYP2C9CYP2C19
SCHEMBL5858677 0.83 ESR1 (0.72) ESR1PLAAALDH1A1CYP1A2CYP2C9
SCHEMBL20880515 0.82 ESR1 (0.64) ESR1PLAAALDH1A1CYP2C9CYP2C19
SCHEMBL20880525 0.82 ESR1 (0.64) ESR1PLAAALDH1A1CYP2C9CYP2C19
SCHEMBL17916294 0.81 ESR1 (0.62) ESR1PLAAL3MBTL1ALDH1A1CYP2C9
SCHEMBL30775444 0.81 ESR1 (1.00) ESR1PLAAMAPK1ALPGPDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563123-B1 NOVEL BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2018-04-25 EP disclosed