SCHEMBL2008454

SCHEMBL2008454

[O]C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)F

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180171 0.97 TSHR (0.39) KDM4ETSHRTDP1
SCHEMBL2634978 0.90 KDM4E (0.42) KDM4ETSHRTDP1
SCHEMBL498059 0.83 KDM4E (0.43) KDM4ETSHRTDP1
SCHEMBL5487202 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL1827978 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL5492824 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL1824897 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL1824498 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL5489726 0.79 TSHR (0.42) KDM4ETSHRTDP1
SCHEMBL1829371 0.79 TSHR (0.42) KDM4ETSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935224-A1 NEW SUBSTITUTED TRIAZOLES AND IMIDAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-28 EP disclosed
EP-2928897-A1 NEW SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-14 EP disclosed
WO-2015150343-A1 SUBSTITUTED 1,3-DITHIOLE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-08 WO disclosed
WO-2015150139-A1 SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-08 WO disclosed
WO-2015150170-A1 SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-08 WO disclosed
WO-2015150138-A1 SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-08 WO disclosed
WO-2015150135-A1 SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-10-08 WO disclosed
EP-2871960-A1 SUBSTITUTED THIADIAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2015-05-20 EP disclosed
WO-2014202751-A1 METHODS FOR CONTROLLING PESTS IN SOYBEAN BASF SE (DE) 2014-12-24 WO disclosed
EP-2802212-A1 HERBICIDAL ISOXAZOLO[5,4-B]PYRIDINES BASF SE (DE) 2014-11-19 EP disclosed
WO-2014095534-A1 NEW SUBSTITUTED TRIAZOLES AND IMIDAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-06-26 WO disclosed
WO-2014095547-A1 NEW SUBSTITUTED TRIAZOLES AND IMIDAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-06-26 WO disclosed
WO-2014095555-A1 NEW SUBSTITUTED TRIAZOLES AND IMIDAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-06-26 WO disclosed
WO-2014086601-A1 NEW SUBSTITUTED 1,4-DITHIINE DERIVATIVES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-06-12 WO disclosed
WO-2014009293-A1 NEW SUBSTITUTED THIADIAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-01-16 WO disclosed
WO-2014009137-A1 SUBSTITUTED THIADIAZOLES AND THEIR USE AS FUNGICIDES BASF SE (DE) 2014-01-16 WO disclosed
WO-2013104561-A1 HERBICIDAL ISOXAZOLO[5,4-B]PYRIDINES BASF SE (DE) 2013-07-18 WO disclosed
WO-2011064188-A1 INSECTICIDAL METHODS USING NITROGEN-CONTAINING HETEROAROMATIC COMPOUNDS BASF SE (DE) 2011-06-03 WO disclosed