SCHEMBL2009434

SCHEMBL2009434

Cc1c(CC(=O)O)c2cc(O)c(F)cc2n1C(=O)C1CCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.40
AKR1C2 P52895 7/20 0.40
PTGS1 P23219 3/20 0.39
PTGS2 P35354 3/20 0.39
PTGDR2 Q9Y5Y4 7/20 0.37
PTGDR Q13258 2/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
HIF1A Q16665 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
TSHR P16473 1/20 0.36
NFKB1 P19838 1/20 0.36
ABCB1 P08183 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
PTGES O14684 1/20 0.35
ABCC3 O15438 1/20 0.35
ABCC4 O15439 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2001558 0.98 AKR1C3 (0.40) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2006034 0.97 AKR1C3 (0.40) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2008025 0.91 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2006804 0.91 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2008035 0.90 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2006014 0.90 AKR1C3 (0.39) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2005949 0.86 PTGS1 (0.45) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2002091 0.86 PTGS1 (0.48) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2004018 0.84 PTGS2 (0.45) AKR1C3AKR1C2PTGS1PTGS2PTGDR2
SCHEMBL2001687 0.84 PTGS1 (0.48) AKR1C3AKR1C2PTGS1PTGS2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7960544-B2 Useful indole compounds IRONWOOD PHARMACEUTICALS, INC. (US) 2011-06-14 US disclosed