SCHEMBL20095954

SCHEMBL20095954

N#Cc1cc(CBr)cc(F)c1Br

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CHKA P35790 1/20 0.31
DAO P14920 1/20 0.31
MAOB P27338 2/20 0.30
MAOA P21397 1/20 0.30
KHK P50053 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411071 0.82 TRPV4 (0.35) TRPV4CYP11B1CYP11B2CHKADAO
SCHEMBL30048138 0.82 TRPV4 (0.35) TRPV4CYP11B1CYP11B2CHKADAO
SCHEMBL24357673 0.79 KDM1A (0.37)
SCHEMBL2651893 0.75 TRPV4 (0.39) TRPV4ESR1ESR2CYP11B1CYP11B2
SCHEMBL17316422 0.75 TRPV4 (0.52) TRPV4
SCHEMBL240133 0.74 TRPV4 (0.57) TRPV4CYP11B1CYP11B2DAOMAOB
SCHEMBL51855 0.74 TRPV4 (0.42) TRPV4CYP11B1CYP11B2CHKADAO
SCHEMBL29413279 0.74 TRPV4 (0.42) TRPV4CYP11B1CYP11B2CHKADAO
SCHEMBL22802432 0.73 TRPV4 (0.41) TRPV4
SCHEMBL22119927 0.72 KHK (0.39) TRPV4ESR1ESR2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018075871-A1 NOVEL ANTIBIOTICS AND METHODS OF USING SAME THE BROAD INSTITUTE, INC. (US) 2018-04-26 WO disclosed