SCHEMBL20101396

SCHEMBL20101396

C/C=C\C=C/Oc1cccc(-c2c(CC(=O)O)cnc3ccccc23)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 14/20 0.43
NR1H3 Q13133 13/20 0.43
PPARG P37231 4/20 0.43
PPARD Q03181 3/20 0.43
PPARA Q07869 3/20 0.43
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16624693 0.80 NR1H2 (0.59) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL16624627 0.78 SMN1; SMN2 (0.55) NR1H2NR1H3ALDH1A1HPGDHTT
SCHEMBL16624697 0.72 MAPT (0.53) NR1H2PPARGALDH1A1HPGDHTT
SCHEMBL16624694 0.71 NR1H2 (0.52) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL16624688 0.71 ALDH1A1 (0.50) ALDH1A1HPGDHTTCYP1A2CYP3A4
SCHEMBL17955245 0.70 NR1H2 (0.51) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL27971255 0.69 KDM4E (0.48) ALDH1A1HPGDHTTNPSR1SMN1; SMN2
SCHEMBL16624731 0.69 NR1H2 (0.44) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL20216017 0.68 NR1H2 (0.49) NR1H2NR1H3PPARGPPARDPPARA
SCHEMBL17954340 0.68 NR1H2 (0.49) NR1H2NR1H3PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052107-B1 ORGANIC COMPOUNDS TO TREAT HEPATITIS B VIRUS NOVARTIS AG (CH) 2018-05-02 EP disclosed