SCHEMBL20101407

SCHEMBL20101407

C=[PH](CC)OCc1ccc2c(c1)OCc1cc(CCc3cccc(CO)c3)ccc1-2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PRF1 P14222 1/20 0.33
ACHE P22303 1/20 0.33
CALM1 P0DP23 1/20 0.33
ROCK2 O75116 13/20 0.32
ROCK1 Q13464 2/20 0.32
AKR1B1 P15121 1/20 0.32
KCNJ1 P48048 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17954207 0.80 PRF1 (0.37) PRF1ACHEROCK2ROCK1AKR1B1
SCHEMBL17954215 0.75 MAOB (0.48) ROCK2
SCHEMBL17954212 0.74 AKR1B1 (0.40) PRF1ACHEROCK2AKR1B1
SCHEMBL20216036 0.72 ROCK2 (0.38) PRF1ACHEROCK2ROCK1AKR1B1
SCHEMBL18165309 0.71 FFAR1 (0.51) AKR1B1
SCHEMBL20788480 0.70 AKR1B1 (0.56) PRF1ACHEROCK2ROCK1AKR1B1
SCHEMBL803505 0.70 KCNJ1 (0.43) ROCK2ROCK1AKR1B1KCNJ1KCNH2
SCHEMBL30529078 0.70 AKR1B1 (0.56) PRF1ACHEROCK2ROCK1AKR1B1
SCHEMBL16624701 0.69 ROCK2 (0.38) ROCK2ROCK1
SCHEMBL17954236 0.69 ROCK2 (0.39) ROCK2ROCK1AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052107-B1 ORGANIC COMPOUNDS TO TREAT HEPATITIS B VIRUS NOVARTIS AG (CH) 2018-05-02 EP disclosed