SCHEMBL20105786

SCHEMBL20105786

Cn1c(=O)[nH]c(=O)c2c1nc(Cn1ccc(N)nc1=O)n2Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.50
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 2/20 0.46
BRDT Q58F21 1/20 0.46
TPH1 P17752 3/20 0.46
TPH2 Q8IWU9 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
ATM Q13315 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 2/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15923850 0.82 GAA (0.56) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL15924216 0.81 MEN1 (0.55) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL15923656 0.76 KMT2A (0.53) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL15924451 0.72 KMT2A (0.58) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL16363970 0.68 ATM (0.55) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL2035525 0.67 F2R (0.48) MEN1KMT2APOLB
SCHEMBL555082 0.66 BRAF (0.72) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL23202390 0.65 MEN1 (0.47) ALDH1A1MEN1KMT2APOLBTPH1
SCHEMBL16076188 0.65 BRDT (0.71) GAAALDH1A1MEN1KMT2APOLB
SCHEMBL22800966 0.65 ALDH1A1 (0.62) GAAALDH1A1MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2951180-B1 2,6,7,8 SUBSTITUTED PURINES AS HDM2 INHIBITORS MERCK SHARP & DOHME (US) 2018-05-02 EP disclosed