SCHEMBL2010730

SCHEMBL2010730

Cc1cc2occ(C(=O)N(C)[C@H](CCNC(=O)c3cccn3C)Cc3ccccc3)c2cc1C

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.58
HCRTR2 O43614 2/20 0.58
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
HRH3 Q9Y5N1 2/20 0.35
KMT2A Q03164 1/20 0.34
MAOB P27338 2/20 0.34
PADI4 Q9UM07 3/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011442 1.00 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2014119 0.90 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL2011116 0.85 HCRTR1 (0.64) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2013106 0.83 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2014644 0.82 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2014998 0.82 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2012749 0.81 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2011090 0.81 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL2015342 0.81 HCRTR1 (0.63) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL13139060 0.80 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed