SCHEMBL20107955

SCHEMBL20107955

CCCCOc1cc(Br)c(F)cc1C(=O)NC(CC)CC

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.50
FAAH O00519 2/20 0.41
HTT P42858 2/20 0.40
RECQL P46063 1/20 0.40
DHODH Q02127 6/20 0.40
TAS1R3 Q7RTX0 2/20 0.39
TAS1R1 Q7RTX1 2/20 0.39
TAS1R2 Q8TE23 1/20 0.38
SCN9A Q15858 1/20 0.38
PKM P14618 1/20 0.38
PPARG P37231 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29816545 0.82 DHODH (0.58) DHODH
SCHEMBL20107945 0.82 DHODH (0.58) DHODH
SCHEMBL28823372 0.82 DHODH (0.58) DHODH
SCHEMBL19684853 0.81 TSHR (0.51)
SCHEMBL19684923 0.81 HTT (0.41) CNR2FAAHHTTRECQLSCN9A
SCHEMBL18021138 0.78 ESR1 (0.51)
SCHEMBL22987098 0.75 SMN1; SMN2 (0.40) HTTRECQL
SCHEMBL12588846 0.75 SCN9A (0.41) FAAHHTTRECQLSCN9A
SCHEMBL20107607 0.75 DHODH (0.47) HTTRECQLDHODH
SCHEMBL20107926 0.74 DHODH (0.53) HTTRECQLDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3532468-B1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AG (DE) 2022-03-23 EP disclosed
WO-2018077923-A1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed