SCHEMBL20108162

SCHEMBL20108162

COC(=O)c1sccc1OC(C)c1ccccc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
PLK1 P53350 6/20 0.43
PLK3 Q9H4B4 4/20 0.43
MEN1 O00255 2/20 0.43
CYP1A2 P05177 1/20 0.43
NEK2 P51955 2/20 0.42
KDM4E B2RXH2 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.39
IKBKE Q14164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30427708 0.88 PLK1 (0.44) PLK1PLK3NEK2
SCHEMBL29453063 0.87 PLK1 (0.51) PLK1PLK3NEK2
SCHEMBL29536039 0.87 PLK1 (0.51) PLK1PLK3NEK2
SCHEMBL3963311 0.87 PLK1 (0.51) PLK1PLK3NEK2
SCHEMBL1370903 0.81 KMT2A (0.51) KMT2APLK1PLK3MEN1CYP1A2
SCHEMBL25267168 0.81 PLK1 (0.49) PLK1PLK3NEK2
SCHEMBL2977455 0.81 PLK1 (0.49) PLK1PLK3NEK2
SCHEMBL30426721 0.81 PLK1 (0.49) PLK1PLK3NEK2
Hydrochloric Acid SCHEMBL3118930 0.80 PLK1 (0.49) PLK1PLK3NEK2
SCHEMBL4777503 0.79 PLK1 (0.49) PLK1PLK3NEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081719-A1 SMALL MOLECULE INHIBITORS OF NEK2 AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2018-05-03 WO disclosed