SCHEMBL20108206

SCHEMBL20108206

CCCCOc1cc(Br)c(F)cc1C(=O)Nc1c(C)ccnc1OC

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 16/20 0.49
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
PDE4D Q08499 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20107602 0.87 DHODH (0.49) DHODH
SCHEMBL20108205 0.86 DHODH (0.66) DHODH
SCHEMBL21853408 0.86 DHODH (0.66) DHODH
SCHEMBL29816492 0.86 DHODH (0.66) DHODH
SCHEMBL20107607 0.83 DHODH (0.47) DHODHHTTRECQLPDE4D
SCHEMBL28953480 0.82 DHODH (0.51) DHODH
SCHEMBL21853424 0.82 DHODH (0.66) DHODH
SCHEMBL21853426 0.82 DHODH (0.66) DHODH
SCHEMBL20107751 0.79 DHODH (0.73) DHODH
SCHEMBL20108244 0.78 DHODH (0.80) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3532468-B1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AG (DE) 2022-03-23 EP disclosed
WO-2018077923-A1 2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH BAYER AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed