SCHEMBL20109733

SCHEMBL20109733

CCN(C)C(=O)c1cccc(CI)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 2/20 0.55
HPGD P15428 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
HSD17B1 P14061 4/20 0.47
HSD17B2 P37059 4/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
RAB9A P51151 1/20 0.45
PPARG P37231 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
PDK2 Q15119 1/20 0.42
ROCK2 O75116 1/20 0.41
PARP1 P09874 2/20 0.40
ALDH1A1 P00352 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20109830 0.88 KMT2A (0.53) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL14117419 0.87 KMT2A (0.58) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL10268480 0.84 KMT2A (0.55) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL1690607 0.81 KMT2A (0.53) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL17790194 0.81 KMT2A (0.53) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL11913144 0.80 HPGD (0.74) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL14039541 0.79 KMT2A (0.50) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL17119847 0.78 HSD17B1 (0.57) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL1196990 0.77 HPGD (0.51) KMT2AMEN1HPGDTDP1HSD17B1
SCHEMBL12806220 0.75 MAOB (0.51) KMT2AMEN1NPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534152-B1 MACROCYCLES AS FACTOR XIA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-02 EP disclosed