SCHEMBL20111520

SCHEMBL20111520

C[C@H]1CCC(C(=O)O)CN1C(=O)c1nccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 7/20 0.47
HCRTR1 O43613 5/20 0.47
PDE2A O00408 1/20 0.41
CCR3 P51677 2/20 0.40
CNR2 P34972 2/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
RCE1 Q9Y256 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20102675 0.91 HCRTR2 (0.47) HCRTR2HCRTR1PDE2ACCR3CNR2
SCHEMBL15064844 0.81 HCRTR1 (0.58) HCRTR2HCRTR1PDE2ACCR3CNR2
SCHEMBL26124986 0.76 HPGD (0.47) HCRTR2KDM4EALDH1A1GAA
SCHEMBL3570468 0.74 HCRTR1 (0.49) HCRTR1PDE2ACCR3ALDH1A1
SCHEMBL3570473 0.74 HCRTR1 (0.49) HCRTR1PDE2ACCR3ALDH1A1
SCHEMBL8986053 0.72 CNR2 (0.48) CNR2RAB9AALDH1A1MAPT
SCHEMBL15064842 0.71 HCRTR1 (0.53) HCRTR2HCRTR1PDE2ACCR3CNR2
SCHEMBL16447712 0.71 HCRTR2 (0.67) HCRTR2HCRTR1
SCHEMBL17724431 0.70 HCRTR2 (0.44) HCRTR2HCRTR1RAB9A
SCHEMBL26123795 0.70 L3MBTL1 (0.50) HCRTR2HCRTR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180121597-A1 Methods to Prepare and Employ Binding Site Models for Modulation of Phosphatase Activity and Selectivity Determination ALLOSTA PHARMACEUTICALS (US) 2018-05-03 US disclosed