SCHEMBL20111649

SCHEMBL20111649

CC(C)(C)C1CCN(S(=O)(=O)C2CCN(C(C)(C)C)CC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.33
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
ACLY P53396 1/20 0.32
EPHX2 P34913 2/20 0.31
DDIT3 P35638 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21732723 0.90 ACLY (0.33) CYP2D6KCNH2HRH3ACLY
SCHEMBL12201520 0.87 EPHX2 (0.39) CYP2D6KCNH2HRH3ACLYEPHX2
SCHEMBL20111712 0.86 ACLY (0.34) CYP2D6KCNH2HRH3ACLYDDIT3
SCHEMBL24477829 0.84 SMYD3 (0.38) CYP2D6KCNH2HRH3ACLYEPHX2
SCHEMBL21732859 0.84 MEN1 (0.39)
SCHEMBL12384633 0.83 EPHX2 (0.44) CYP2D6KCNH2HRH3ACLYEPHX2
SCHEMBL21732864 0.80 ACLY (0.32) ACLYEPHX2
SCHEMBL2706991 0.80 CYP2D6 (0.38) CYP2D6KCNH2HRH3EPHX2
SCHEMBL21732954 0.79 SMYD3 (0.31)
SCHEMBL12040228 0.79 EPHX2 (0.35) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10961238-B2 Modulators of hedgehog (Hh) signaling pathway E-THERAPEUTICS PLC (GB) 2021-03-30 US disclosed
US-20200055847-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY E-THERAPEUTICS PLC (GB) 2020-02-20 US disclosed
WO-2018078360-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY E-THERAPEUTICS PLC (GB) 2018-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10961238-B2 Modulators of hedgehog (Hh) signaling pathway SHH, GLI1, SMO CYP2D6 4442/4885KCNH2 4799/4885HRH3 901/4885
US-20200055847-A1 MODULATORS OF HEDGEHOG (HH) SIGNALLING PATHWAY SHH, GLI1, SMO CYP2D6 4378/4885KCNH2 4785/4885HRH3 766/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.