SCHEMBL20113745

SCHEMBL20113745

CC(C)(O)C#Cc1nc(Cl)n(Cc2ccc(F)cc2)c1C(=O)NCC1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
KCNH2 Q12809 1/20 0.39
CACNA1I Q9P0X4 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CNR1 P21554 6/20 0.38
CNR2 P34972 6/20 0.38
FAAH O00519 2/20 0.38
MAP3K14 Q99558 1/20 0.38
MAPT P10636 1/20 0.38
HTR4 Q13639 1/20 0.37
RIPK1 Q13546 1/20 0.37
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC6 Q9UBN7 2/20 0.36
MLYCD O95822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20113514 0.92 NPC1 (0.46) RAB9ANPC1KCNH2CACNA1IKMT2A
SCHEMBL20113478 0.91 PTGER4 (0.43) KCNH2CACNA1IHDAC6MLYCD
SCHEMBL20113518 0.91 NPC1 (0.41) RAB9ANPC1KCNH2CACNA1ICNR2
SCHEMBL16305010 0.91 PTGER4 (0.44) MEN1KMT2AMAP3K14HTR4RIPK1
SCHEMBL18626493 0.91 PTGER4 (0.44) MEN1KMT2AMAP3K14HTR4RIPK1
SCHEMBL20113498 0.88 HDAC6 (0.38) KCNH2CACNA1IMEN1KMT2ACNR1
SCHEMBL20113509 0.86 PTGER4 (0.44) KCNH2CACNA1IHDAC6MLYCD
SCHEMBL16305011 0.83 PTGER4 (0.43) KCNH2CACNA1IMEN1KMT2AMAP3K14
SCHEMBL18626441 0.83 PTGER4 (0.43) KCNH2CACNA1IMEN1KMT2AMAP3K14
SCHEMBL20113520 0.83 PTGER4 (0.42) KCNH2CACNA1IHDAC6MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3009426-B1 4-ALKYNYL IMIDAZOLE DERIVATIVE AND MEDICINE COMPRISING SAME AS ACTIVE INGREDIENT KAKEN PHARMA CO LTD (JP) 2018-05-02 EP disclosed