SCHEMBL20113478

SCHEMBL20113478

CC(C)(O)C#Cc1nc(Cl)n(Cc2ccc(C(F)(F)F)cc2)c1C(=O)NCC1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.43
MDM2 Q00987 8/20 0.42
HDAC6 Q9UBN7 2/20 0.39
MLYCD O95822 1/20 0.39
GSK3B P49841 1/20 0.38
RORC P51449 3/20 0.37
KCNH2 Q12809 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
GLS O94925 1/20 0.36
NAPEPLD Q6IQ20 1/20 0.36
CETP P11597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20113509 0.95 PTGER4 (0.44) PTGER4MDM2HDAC6MLYCDGSK3B
SCHEMBL20113520 0.92 PTGER4 (0.42) PTGER4MDM2HDAC6MLYCDGSK3B
SCHEMBL20113745 0.91 RAB9A (0.42) HDAC6MLYCDKCNH2CACNA1I
SCHEMBL16304056 0.91 PTGER4 (0.41) PTGER4MDM2HDAC6MLYCDGSK3B
SCHEMBL17684492 0.91 PTGER4 (0.54) PTGER4MDM2GSK3BRORCKCNH2
SCHEMBL16305068 0.91 PTGER4 (0.54) PTGER4MDM2GSK3BRORCKCNH2
SCHEMBL16304872 0.91 AGTR2 (0.42) PTGER4MDM2HDAC6MLYCDGSK3B
SCHEMBL20113514 0.91 NPC1 (0.46) KCNH2CACNA1IGLS
SCHEMBL20113498 0.90 HDAC6 (0.38) HDAC6MLYCDKCNH2CACNA1IGLS
SCHEMBL17684823 0.90 PTGER4 (0.45) PTGER4MDM2GSK3BRORCKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3009426-B1 4-ALKYNYL IMIDAZOLE DERIVATIVE AND MEDICINE COMPRISING SAME AS ACTIVE INGREDIENT KAKEN PHARMA CO LTD (JP) 2018-05-02 EP disclosed