SCHEMBL20116207

SCHEMBL20116207

COc1ccc(C(=O)CBr)cc1OC(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.61
MAPT P10636 4/20 0.50
TSHR P16473 2/20 0.50
CTNNB1 P35222 2/20 0.50
WNT3A P56704 2/20 0.50
GSK3B P49841 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA6 P23280 1/20 0.47
CA7 P43166 1/20 0.47
TPMT P51580 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
ALDH1A1 P00352 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL426444 0.87 TSHR (0.63) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL29620831 0.87 TSHR (0.63) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL21611281 0.87 PDE4B (0.48) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL661011 0.86 PDE4B (0.62) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL6060600 0.84 PDE4B (0.60) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL4277719 0.81 MAPK1 (0.59) PDE4BMAPTTSHRCYP1A2CYP3A4
SCHEMBL661271 0.81 ALDH1A1 (0.56) PDE4BMAPTTSHRCYP1A2CYP3A4
SCHEMBL3924278 0.81 CA12 (0.73) PDE4BTSHRCYP1A2CYP3A4CYP2C9
SCHEMBL9204477 0.81 KDM4E (0.54) PDE4BMAPTTSHRCTNNB1WNT3A
SCHEMBL25139577 0.80 MEN1 (0.62) PDE4BMAPTTSHRCTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed