SCHEMBL20116283

SCHEMBL20116283

Cc1ccc2cnn(C3CNC3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KHK P50053 5/20 0.42
KMO O15229 1/20 0.40
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
KDM1A O60341 1/20 0.37
CHRM2 P08172 3/20 0.36
CHRM1 P11229 3/20 0.36
CHRM3 P20309 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR1A P08908 1/20 0.36
HTR1B P28222 1/20 0.36
HTR1F P30939 1/20 0.36
CYP11B2 P19099 1/20 0.34
SCD O00767 2/20 0.34
KDM5A P29375 1/20 0.34
PDE2A O00408 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15830331 0.88 KDM1A (0.44) KHKKMOHTR2AHTR2CHTR2B
SCHEMBL13432160 0.85 KMO (0.43) KMOKDM1ACHRM2CHRM1CHRM3
SCHEMBL15830291 0.85 KDM1A (0.51) KHKKMOKDM1ACHRM2CHRM1
SCHEMBL17678157 0.83 KMO (0.41) KMOKDM1ACHRM2CHRM1CHRM3
SCHEMBL26811385 0.81 HTR2A (0.44) KHKHTR2AHTR2CHTR2BCHRNB2
SCHEMBL20116574 0.81 PDE1B (0.40) KMOCHRM2CHRM1CHRM3HTR1A
SCHEMBL20116866 0.81 KMO (0.43) KHKKMOCHRM2CHRM1CHRM3
SCHEMBL26997309 0.81 KDM5A (0.39) KHKCHRNB2CHRNA4HTR1AHTR1B
SCHEMBL22358062 0.81 SCD (0.39) KHKHTR2AHTR2CHTR2BHTR1A
SCHEMBL26811388 0.81 HTR2C (0.46) HTR2AHTR2CHTR2BCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed