SCHEMBL20116289

SCHEMBL20116289

Cc1ccn2cnc(I)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TP53 P04637 1/20 0.34
KDM4E B2RXH2 5/20 0.33
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
APOBEC3A P31941 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
ALDH1A1 P00352 2/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
FGFR1 P11362 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17815221 0.80 CCR1 (0.37) CCR1CCR5CCR8SMN1; SMN2TP53
SCHEMBL25044254 0.80 IDO1 (0.30)
SCHEMBL22358029 0.77
SCHEMBL20116290 0.74 TP53 (0.33) CCR1CCR5CCR8SMN1; SMN2TP53
SCHEMBL21893418 0.74 KDM4E (0.37) CCR1CCR5CCR8SMN1; SMN2TP53
SCHEMBL24657617 0.74 TP53 (0.33) CCR1CCR5CCR8SMN1; SMN2TP53
SCHEMBL21358993 0.73 KLKB1 (0.34) CCR1CCR5CCR8SMN1; SMN2TP53
Hydrochloric Acid SCHEMBL28568645 0.73 IKBKB (0.42) CCR1CCR5CCR8SMN1; SMN2TP53
Hydrochloric Acid SCHEMBL21355066 0.72 KLKB1 (0.34) CCR1CCR5CCR8SMN1; SMN2TP53
SCHEMBL19641513 0.72 KDM4E (0.40) SMN1; SMN2KDM4EALDH1A1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed