SCHEMBL20116645

SCHEMBL20116645

COc1ccc(-c2noc(C3CCN(C(=O)CI)CC3)n2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.58
TSHR P16473 2/20 0.58
MEN1 O00255 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C9 P11712 1/20 0.58
CYP2C19 P33261 1/20 0.58
KMT2A Q03164 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
LMNA P02545 2/20 0.57
USP2 O75604 1/20 0.57
SMO Q99835 1/20 0.57
ALOX15 P16050 1/20 0.52
MAPK1 P28482 1/20 0.52
TLR9 Q9NR96 1/20 0.51
TLR8 Q9NR97 1/20 0.51
TLR7 Q9NYK1 1/20 0.51
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116646 0.91 HTT (0.59) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20116204 0.90 HTT (0.58) HTTTSHRMEN1CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL30506238 0.89 HTT (0.58) HTTTSHRMEN1CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL20660764 0.89 HTT (0.58) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20116341 0.86 HTT (0.57) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20116121 0.86 TSHR (0.71) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20660946 0.86 SMO (0.56) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20116343 0.84 TSHR (0.65) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20116344 0.84 SMO (0.53) HTTTSHRMEN1CYP3A4CYP2C9
SCHEMBL20117193 0.83 SMO (0.55) HTTTSHRMEN1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed