SCHEMBL20116740

SCHEMBL20116740

CC(C)(C)OC(=O)N1CC(n2ncc3ccc(-c4noc(C5CCN(C=O)CC5)n4)cc32)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.43
GPR119 Q8TDV5 3/20 0.43
HDAC4 P56524 3/20 0.41
HDAC6 Q9UBN7 2/20 0.41
NR1H4 Q96RI1 1/20 0.40
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TUBB4A P04350 3/20 0.39
TUBB P07437 3/20 0.39
TUBA3C P0DPH7 3/20 0.39
TUBA1B P68363 3/20 0.39
TUBA4A P68366 3/20 0.39
TUBB4B P68371 3/20 0.39
TUBB3 Q13509 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20116621 0.93 GPR119 (0.50) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20676227 0.90 GPR119 (0.48) SMOGPR119HDAC4HDAC6MEN1
SCHEMBL20116075 0.89 GPR119 (0.48) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20116681 0.88 SMO (0.45) SMONR1H4MEN1CYP3A4CYP2C9
SCHEMBL22358247 0.88 GPR119 (0.54) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20116323 0.86 GPR119 (0.52) SMOGPR119HDAC4HDAC6TUBB4A
SCHEMBL22358260 0.85 GPR119 (0.49) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20116418 0.85 GPR119 (0.49) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20676322 0.85 GPR119 (0.49) SMOGPR119HDAC4HDAC6TSHR
SCHEMBL20116966 0.85 GPR119 (0.49) SMOGPR119HDAC4HDAC6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed