SCHEMBL20117306

SCHEMBL20117306

Cc1cnc2c(C)nn(C)c2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
CCR1 P32246 3/20 0.43
CCR5 P51681 3/20 0.43
CCR8 P51685 3/20 0.43
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PSMD14 O00487 1/20 0.35
COPS5 Q92905 1/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
HDAC6 Q9UBN7 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
PDE10A Q9Y233 1/20 0.32
CYP1A2 P05177 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
PARP1 P09874 1/20 0.31
MAPK1 P28482 1/20 0.31
GRM4 Q14833 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27259309 0.82 ADORA2A (0.42) ADORA2AADORA2BCCR1CCR5CCR8
SCHEMBL17674371 0.82 HSD17B10 (0.43) ADORA2AADORA2BCCR1CCR5CCR8
SCHEMBL30968108 0.82 CCR1 (0.39) ADORA2AADORA2BCCR1CCR5CCR8
SCHEMBL30506328 0.82 HSD17B10 (0.43) ADORA2AADORA2BCCR1CCR5CCR8
SCHEMBL20116648 0.80 ADORA2A (0.40) ADORA2AADORA2BKDM4EALDH1A1HRH4
SCHEMBL17678134 0.78 ADORA2A (0.39) ADORA2AADORA2BKDM4EALDH1A1SLC22A12
SCHEMBL5363077 0.78 ADORA2A (0.41) ADORA2AADORA2B
Ammonia Solution, Strong SCHEMBL29161534 0.76 ADORA2A (0.39) ADORA2AADORA2B
SCHEMBL20116494 0.73 SLC22A12 (0.35) ADORA2AADORA2BSLC22A12MAPK1SPR
SCHEMBL20661130 0.73 SLC22A12 (0.35) ADORA2AADORA2BHDAC6SLC22A12SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021254493-A1 CYCLIC COMPOUND HAVING ANTI-TUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2021-12-23 WO disclosed
WO-2019209948-A9 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-01-02 WO disclosed
WO-2019018795-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2019-01-24 WO disclosed
WO-2018081167-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS (US) 2018-05-03 WO disclosed