SCHEMBL30968108

SCHEMBL30968108

Cc1cnc2c(Br)nn(C)c2c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.39
CCR5 P51681 3/20 0.39
CCR8 P51685 3/20 0.39
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PSMD14 O00487 1/20 0.33
COPS5 Q92905 1/20 0.33
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117306 0.82 ADORA2A (0.47) CCR1CCR5CCR8ADORA2AADORA2B
SCHEMBL30506328 0.74 HSD17B10 (0.43) CCR1CCR5CCR8ADORA2AADORA2B
SCHEMBL17674371 0.74 HSD17B10 (0.43) CCR1CCR5CCR8ADORA2AADORA2B
SCHEMBL20951908 0.72 PSMD14 (0.43) KDM4EALDH1A1PSMD14
SCHEMBL14074978 0.68 SSTR4 (0.38) CCR1CCR5CCR8ADORA2AKDM4E
SCHEMBL27259309 0.67 ADORA2A (0.42) CCR1CCR5CCR8ADORA2AADORA2B
SCHEMBL30791898 0.66 HSD17B10 (0.42) KDM4EALDH1A1
SCHEMBL20741029 0.66 HSD17B10 (0.42) KDM4EALDH1A1
SCHEMBL15342706 0.66 SMN1; SMN2 (0.32)
SCHEMBL33526224 0.66 HSD17B10 (0.42) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118239959-A Cyclopropane TLR7 and 8 inhibitor and preparation method and application thereof 上海深势唯思科技有限责任公司 2024-06-25 CN disclosed