SCHEMBL20117432

SCHEMBL20117432

CC1CCCN1c1nc(C(N)=O)cc(-c2ccc(Oc3ccc(OC(F)(F)F)cc3)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 18/20 0.52
KDM4E B2RXH2 2/20 0.51
ALDH1A1 P00352 2/20 0.51
GAA P10253 2/20 0.51
HPGD P15428 2/20 0.51
TP53 P04637 1/20 0.51
FPR2 P25090 6/20 0.49
TSHR P16473 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16013421 0.89 SCN9A (0.60) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL16012982 0.89 SCN9A (0.60) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL3717819 0.84 SCN9A (0.51) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL3727036 0.84 SCN9A (0.51) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL3727334 0.84 SCN9A (0.51) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL19956218 0.84 JAK2 (0.42) SCN9AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL19956223 0.84 FPR2 (0.66) SCN9AFPR2
SCHEMBL19956217 0.81 SCN9A (0.51) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL1734370 0.80 KDM4E (0.74) SCN9AKDM4EALDH1A1GAAHPGD
SCHEMBL16012691 0.75 SCN9A (0.83) SCN9AFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964639-B1 PYRIMIDINE CARBOXAMIDES AS SODIUM CHANNEL BLOCKERS PURDUE PHARMA LP (US) 2018-05-02 EP disclosed