SCHEMBL20117852

SCHEMBL20117852

Cc1ccccc1Cc1cccn1-c1ccc(C(N)=O)c(NC2CCCCC2)c1

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90B1 P14625 2/20 0.69
HSP90AA1 P07900 16/20 0.45
HSP90AB1 P08238 3/20 0.45
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
TRAP1 Q12931 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20117851 0.92 HSP90B1 (0.82) HSP90B1HSP90AA1HSP90AB1
SCHEMBL20117712 0.89 HSP90B1 (0.69) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117836 0.88 HSP90B1 (0.66) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117732 0.87 HSP90B1 (0.65) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117738 0.83 HSP90B1 (0.63) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117787 0.83 HSP90B1 (0.60) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117729 0.82 HSP90B1 (0.60) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117975 0.82 HSP90B1 (0.60) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117976 0.82 HSP90B1 (0.60) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR
SCHEMBL20117688 0.82 HSP90B1 (0.60) HSP90B1HSP90AA1HSP90AB1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081814-A1 GRP94 SELECTIVE INHIBITORS AND USES THEREOF UNIVERSITY OF KANSAS (US) 2018-05-03 WO disclosed