SCHEMBL20118186

SCHEMBL20118186

CC1C[C@]2(CC[C@@H](NC(=O)c3cnn4cccnc34)CC2)C(=O)N1Cc1ccc(F)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
PKM P14618 1/20 0.46
TNKS O95271 1/20 0.43
IRAK4 Q9NWZ3 2/20 0.43
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
NTRK1 P04629 8/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
JAK2 O60674 4/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
PDE2A O00408 1/20 0.40
BMPR1B O00238 1/20 0.40
BMPR1A P36894 1/20 0.40
TGFBR1 P36897 1/20 0.40
ACVRL1 P37023 1/20 0.40
ACVR1 Q04771 1/20 0.40
HSD11B1 P28845 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20185045 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL18216445 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL18208327 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL20185038 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL18208323 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL20185046 0.86 KDM4E (0.46) KDM4EHSD17B10TNKSIRAK4
SCHEMBL20118061 0.86 KDM4E (0.47) KDM4EHSD17B10PKMTNKSIRAK4
SCHEMBL20118060 0.86 KDM4E (0.47) KDM4EHSD17B10PKMTNKSIRAK4
SCHEMBL20118240 0.86 KDM4E (0.47) KDM4EHSD17B10PKMTNKSIRAK4
SCHEMBL18208502 0.79 IRAK4 (0.49) KDM4EHSD17B10TNKSIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018078009-A1 AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-03 WO disclosed