SCHEMBL20119686

SCHEMBL20119686

CCN1CCc2cc(C(=O)NS(=O)(=O)C3(C)CC3)ccc2C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.44
HDAC8 Q9BY41 2/20 0.44
PRMT5 O14744 10/20 0.42
WDR77 Q9BQA1 10/20 0.42
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC3 O15379 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20119182 0.85 HDAC6 (0.46) HDAC6HDAC8HDAC1HDAC3
SCHEMBL20173798 0.82 HDAC6 (0.44) HDAC6HDAC8HDAC1HDAC3
SCHEMBL10120332 0.82 HDAC6 (0.62) HDAC6HDAC8HDAC1HDAC3
SCHEMBL10120344 0.77 HDAC6 (0.56) HDAC6HDAC8HDAC1HDAC3
SCHEMBL20178641 0.75 ALDH1A1 (0.51) HDAC6HDAC8ITGB3ITGA2B
SCHEMBL10120339 0.75 HDAC6 (0.64) HDAC6HDAC8HDAC1HDAC3
SCHEMBL20178679 0.74 ACACB (0.59) HDAC6HDAC8PRMT5WDR77
SCHEMBL10120343 0.74 HDAC6 (0.63) HDAC6HDAC8HDAC1HDAC3
SCHEMBL10120349 0.74 HDAC6 (0.59) HDAC6HDAC8HDAC1HDAC3
SCHEMBL10104761 0.72 HDAC6 (0.57) HDAC6HDAC8PRMT5WDR77HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018081285-A1 UREA-CONTAINING ISOXAZOLE DERIVATIVES AS FXR AGONISTS AND METHODS OF USE THEREOF ENANTA PHARMACEUTICALS, INC. (US) 2018-05-03 WO disclosed