SCHEMBL20121087

SCHEMBL20121087

COC(=O)c1cc2ccc(OC)nc2n1CC1CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
KDM2B Q8NHM5 7/20 0.42
MTNR1A P48039 7/20 0.40
MTNR1B P49286 7/20 0.40
PIK3CA P42336 1/20 0.38
PADI4 Q9UM07 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31215258 0.93 ROCK2 (0.44) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18969559 0.93 ROCK2 (0.44) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18940586 0.89 ROCK2 (0.43) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18960744 0.89 ROCK2 (0.42) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18938869 0.86 ROCK2 (0.45) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18938861 0.85 ROCK2 (0.47) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL29641293 0.85 ROCK2 (0.47) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL18938863 0.84 ROCK2 (0.44) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL29850606 0.84 ROCK2 (0.44) ROCK2ROCK1KDM2BMTNR1AMTNR1B
SCHEMBL19359607 0.83 ROCK2 (0.45) ROCK2ROCK1MTNR1AMTNR1BPADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963448-B2 Bicyclic inhibitors of PAD4 PADLOCK THERAPEUTICS, INC. (US) 2018-05-08 US disclosed