SCHEMBL20121186

SCHEMBL20121186

Cc1ccc(Nc2c(-c3ccc(F)cc3)nc3n2CCN(C(=O)C(C)(N)Cc2ccc(F)cc2)C3)cc1

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.81
CYP3A4 P08684 1/20 0.45
TGFBR1 P36897 2/20 0.37
PDK2 Q15119 1/20 0.37
CSNK1D P48730 3/20 0.36
CSNK1E P49674 3/20 0.36
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2068778 1.00 KCNH2 (0.81) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL15760160 0.98 KCNH2 (0.77) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL15750535 0.92 KCNH2 (0.78) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL15340406 0.91 KCNH2 (0.83) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL2068305 0.91 KCNH2 (0.83) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL1049719 0.91 KCNH2 (0.83) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL15760177 0.90 KCNH2 (0.78) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL2068261 0.89 KCNH2 (1.00) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL20121564 0.89 KCNH2 (0.74) KCNH2CYP3A4TGFBR1PDK2CSNK1D
SCHEMBL2068863 0.89 KCNH2 (0.79) KCNH2CYP3A4TGFBR1PDK2CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed