SCHEMBL20121564

SCHEMBL20121564

Cc1ccc(Nc2c(-c3ccc(F)cc3)nc3n2CCN(C(=O)[C@@](N)(O)Cc2ccc(N)cc2)C3)cc1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.74
CYP3A4 P08684 2/20 0.44
CSNK1D P48730 3/20 0.36
CSNK1E P49674 3/20 0.36
TGFBR1 P36897 2/20 0.36
PDK2 Q15119 1/20 0.35
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15760160 0.92 KCNH2 (0.77) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL2068778 0.89 KCNH2 (0.81) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL15750535 0.89 KCNH2 (0.78) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL20121186 0.89 KCNH2 (0.81) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL20121535 0.89 KCNH2 (0.80) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL2068261 0.85 KCNH2 (1.00) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL12952248 0.85 KCNH2 (0.75) KCNH2CYP3A4
SCHEMBL2069056 0.84 KCNH2 (0.84) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL1049719 0.84 KCNH2 (0.83) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1
SCHEMBL15340406 0.84 KCNH2 (0.83) KCNH2CYP3A4CSNK1DCSNK1ETGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed