SCHEMBL20121548

SCHEMBL20121548

O=C(CCc1ccc(F)cc1)N1CCn2c(nc(-c3ccc(F)cc3)c2Nc2ccc(Cl)c(F)c2)C1

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.80
CYP3A4 P08684 1/20 0.42
KCNK3 O14649 1/20 0.40
MLNR O43193 1/20 0.39
P2RX7 Q99572 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12952198 0.96 KCNH2 (0.74) KCNH2CYP3A4KCNK3MLNRP2RX7
SCHEMBL12952175 0.96 KCNH2 (0.76) KCNH2CYP3A4KCNK3P2RX7MEN1
SCHEMBL20121545 0.95 KCNH2 (0.75) KCNH2CYP3A4KCNK3MLNRP2RX7
SCHEMBL20121543 0.94 KCNH2 (0.71) KCNH2CYP3A4KCNK3MLNR
SCHEMBL20121599 0.92 KCNH2 (0.68) KCNH2CYP3A4MLNR
SCHEMBL12951888 0.91 KCNH2 (0.82) KCNH2CYP3A4KCNK3P2RX7MEN1
SCHEMBL1051508 0.91 KCNH2 (0.81) KCNH2CYP3A4KCNK3P2RX7MEN1
SCHEMBL12951891 0.91 KCNH2 (0.81) KCNH2CYP3A4KCNK3P2RX7
SCHEMBL20121610 0.90 KCNH2 (0.70) KCNH2CYP3A4MLNR
SCHEMBL2071054 0.90 KCNH2 (0.75) KCNH2CYP3A4P2RX7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9963454-B2 Compounds and compositions for the treatment of parasitic disease NOVARTIS AG (CH) 2018-05-08 US disclosed